SCHEMBL8563386

SCHEMBL8563386

CNC(=O)[C@H]1CNc2ccccc2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
EPHX2 P34913 1/20 0.37
SMYD3 Q9H7B4 1/20 0.36
MMP3 P08254 4/20 0.33
BRD4 O60885 3/20 0.33
CREBBP Q92793 3/20 0.33
MMP1 P03956 3/20 0.33
MMP2 P08253 3/20 0.33
MMP9 P14780 3/20 0.33
MMP8 P22894 3/20 0.33
KCNH2 Q12809 1/20 0.33
EP300 Q09472 1/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563390 1.00 GAA (0.40) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL8563383 1.00 GAA (0.40) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL29036196 0.80 MAPT (0.46) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL18955109 0.80 BACE1 (0.44) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL6186463 0.79 MAPT (0.58) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL6419902 0.77 GAA (0.43) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL30146036 0.77 GAA (0.65) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL13610792 0.77 GAA (0.65) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL26780527 0.77 GAA (0.44) GAAMAPTHPGDMTNR1AMTNR1B
SCHEMBL26783406 0.77 GAA (0.40) GAAMAPTHPGDMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed