SCHEMBL8563772

SCHEMBL8563772

CS(=O)(=O)c1ccc2c(c1)C(=O)CC1(CCN(C3CCc4cc(C#N)ccc4C3)CC1)O2

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.58
EPHX2 P34913 4/20 0.46
EPHX1 P07099 2/20 0.46
CYP11B2 P19099 1/20 0.44
HTR2A P28223 2/20 0.42
DRD2 P14416 1/20 0.40
KCNJ1 P48048 1/20 0.40
SCN5A Q14524 1/20 0.39
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA7 P43166 3/20 0.38
CA9 Q16790 3/20 0.38
ATM Q13315 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8831738 0.89 KCNH2 (0.72) KCNH2CYP11B2HTR2AKCNJ1
SCHEMBL8831813 0.89 KCNH2 (0.72) KCNH2CYP11B2HTR2AKCNJ1
SCHEMBL7388074 0.89 KCNH2 (0.72) KCNH2CYP11B2HTR2AKCNJ1
Hydrochloric Acid SCHEMBL9227313 0.88 KCNH2 (0.71) KCNH2CYP11B2HTR2AKCNJ1
Hydrochloric Acid SCHEMBL7359216 0.88 KCNH2 (0.71) KCNH2CYP11B2HTR2AKCNJ1
Hydrochloric Acid SCHEMBL9227094 0.88 KCNH2 (0.71) KCNH2CYP11B2HTR2AKCNJ1
Hydrochloric Acid SCHEMBL6369601 0.87 KCNH2 (0.70) KCNH2CYP11B2HTR2AKCNJ1
SCHEMBL8569281 0.87 KCNH2 (0.62) KCNH2EPHX2EPHX1CYP11B2HTR2A
SCHEMBL8804765 0.86 KCNH2 (0.53) KCNH2EPHX2EPHX1CYP11B2HTR2A
Hydrochloric Acid SCHEMBL8806196 0.85 KCNH2 (0.52) KCNH2EPHX2EPHX1CYP11B2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP claimed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP claimed
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed