SCHEMBL8564825

SCHEMBL8564825

Clc1ccc2[nH][c]nc2c1-c1ccc2ccccc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.37
FABP3 P05413 1/20 0.36
FABP4 P15090 1/20 0.36
FABP5 Q01469 1/20 0.36
CYP1A2 P05177 1/20 0.36
ALOX15 P16050 1/20 0.35
PTGES O14684 1/20 0.35
FASN P49327 1/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
TRPA1 O75762 1/20 0.34
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
NISCH Q9Y2I1 1/20 0.33
PDE9A O76083 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563998 0.85 IKBKB (0.36) IKBKBFABP3FABP4FABP5CYP1A2
SCHEMBL8564792 0.80 RAC1 (0.42) IKBKBNISCHMAPK10
SCHEMBL8564036 0.75 TYMP (0.40) CYP1A2PTGESNISCHCYP2A6
SCHEMBL8566061 0.73 HTR2B (0.49) CYP1A2CYP11B1CYP11B2CYP1A1CYP1B1
SCHEMBL10832750 0.68 MEN1 (0.30)
SCHEMBL28514503 0.68 HPGD (0.33) FASNESR1ESR2
SCHEMBL3103036 0.65 NQO2 (0.43) ESR1ESR2
SCHEMBL29647703 0.65 CYP1A2 (0.58) CYP1A2CYP11B1CYP11B2CYP1A1CYP1B1
SCHEMBL21076148 0.64 AHR (0.64) CYP11B1CYP11B2CYP1B1CYP17A1CYP19A1
SCHEMBL28144887 0.64 IKBKB (0.43) IKBKBFABP3FABP4FABP5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed