SCHEMBL8565414

SCHEMBL8565414

CC[C](C)Cc1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.56
ESR1 P03372 2/20 0.54
CYP19A1 P11511 2/20 0.54
CHRNB2 P17787 3/20 0.50
CHRNA4 P43681 3/20 0.50
CYP1A2 P05177 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2D6 P10635 1/20 0.47
ALDH1A1 P00352 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
FDPS P14324 1/20 0.46
CHRNA7 P36544 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682021 0.82 NAPRT (0.62) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL8915193 0.79 NAPRT (0.65) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL30917345 0.79 NAPRT (0.65) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL8737617 0.78 NAPRT (0.58) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL48669 0.78 NAPRT (0.69) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL25905487 0.78 NAPRT (0.58) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL29611658 0.78 NAPRT (0.69) NAPRTESR1CYP19A1CHRNB2CHRNA4
SCHEMBL7417227 0.78 CYP1A2 (0.59) NAPRTESR1CYP19A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL1978920 0.77 NAPRT (0.67) NAPRTESR1CYP19A1CYP1A2CYP3A4
SCHEMBL10744051 0.76 NAPRT (0.55) NAPRTESR1CYP19A1CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880524-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS Boehringer Ingelheim Pharma KG (DE) 1998-12-02 EP disclosed
WO-1998003511-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-01-29 WO disclosed