SCHEMBL8566833

SCHEMBL8566833

Clc1cccc2n[c]n(Cl)c12

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.41
PSMB8 P28062 2/20 0.38
CYP1A2 P05177 1/20 0.31
CYP2A6 P11509 1/20 0.31
GUSB P08236 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7815243 0.78 PRMT5 (0.47) PRMT5PSMB8CYP1A2CYP2A6PARP1
SCHEMBL17186937 0.74 PRMT5 (0.40) PRMT5PSMB8
SCHEMBL5000469 0.72 PRMT5 (0.41) PRMT5PSMB8
SCHEMBL10832749 0.68 GRM2 (0.36) CYP1A2CYP2A6PARP1
SCHEMBL3282387 0.64 KDM4E (0.49) PRMT5PSMB8
SCHEMBL14717084 0.62 MEN1 (0.35)
SCHEMBL1359399 0.61 PSMB8 (0.41) PRMT5PSMB8CYP1A2CYP2A6GUSB
SCHEMBL2274904 0.60 PSMB8 (0.38) PRMT5PSMB8PARP1
SCHEMBL21187468 0.60 DPP4 (0.51) PRMT5PSMB8
SCHEMBL10775894 0.60 DPP4 (0.51) PRMT5PSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814646-A TREATING THE PROGRESSION OF ALZHEIMER'S DISEASE, BRAIN DISORDERS ELI LILLY AND COMPANY (US) 1998-09-29 US disclosed