SCHEMBL8567572

SCHEMBL8567572

N#Cc1ccc(CCN2CCC3(CC2)CC(=O)c2cc4[nH]c(=O)[nH]c4cc2O3)cc1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.55
HDAC3 O15379 2/20 0.45
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC10 Q969S8 2/20 0.45
HDAC11 Q96DB2 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45
KCNH2 Q12809 3/20 0.44
KCNJ1 P48048 2/20 0.44
ADRA1D P25100 3/20 0.42
ADRA1A P35348 3/20 0.42
ADRA1B P35368 3/20 0.42
DRD2 P14416 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8567680 0.99 HTR2A (0.54) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL9854607 0.87 HDAC3 (0.57) HTR2AHDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8566808 0.86 HDAC3 (0.56) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL8566373 0.85 HTR2A (0.58) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL8563152 0.85 HTR2A (0.51) HTR2AHDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8569582 0.85 HTR2A (0.57) HTR2AHDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8566387 0.85 HTR2A (0.59) HTR2AHDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8567003 0.84 HTR2A (0.51) HTR2AHDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8562002 0.83 HTR2A (0.45) HTR2AKCNH2KCNJ1ADRA1DADRA1A
SCHEMBL8565543 0.81 HTR2A (0.51) HTR2AHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP claimed