SCHEMBL856798

SCHEMBL856798

CC[C@H]1CCc2c(ncnc2N2CCOc3ccc(-c4cnc5nc(N(C)C(=O)O)[nH]c5c4)cc3C2)C1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.34
KIT P10721 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
TBK1 Q9UHD2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL856549 0.92 PIK3CA (0.33) PIK3CA
SCHEMBL3717364 0.88 PIK3CA (0.34) PIK3CAKITKDM4ETSHRHTT
SCHEMBL858635 0.87 PIK3CA (0.35) PIK3CAKITKDM4ETSHRHTT
SCHEMBL3767906 0.87 KDM4E (0.34) PIK3CAKITKDM4ETSHRHTT
SCHEMBL7859249 0.85 PIK3CA (0.33) PIK3CAKITKDM4ETSHRHTT
SCHEMBL15522787 0.84 PIK3CA (0.35) PIK3CA
SCHEMBL3762761 0.84 KDM4E (0.32) PIK3CAKITKDM4ETSHRHTT
SCHEMBL3768247 0.84 KDM4E (0.32) PIK3CAKITKDM4ETSHRHTT
SCHEMBL861157 0.83 PIK3CA (0.34) PIK3CAKITKDM4ETSHRHTT
SCHEMBL859124 0.83 PIK3CA (0.36) PIK3CAKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432779-A1 BENZOXAZEPINES BASED P13K/MT0R INHIBITORS AGAINST PROLIFERATIVE DISEASES Exelixis, Inc. (US) 2012-03-28 EP disclosed