SCHEMBL8568569

SCHEMBL8568569

COc1ccc(C(=O)Cl)c2[nH]c(C3CC3)nc12

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.56
PDE4B Q07343 2/20 0.56
PDE4C Q08493 2/20 0.56
PDE4D Q08499 2/20 0.56
PARP1 P09874 2/20 0.43
PBK Q96KB5 9/20 0.41
HTR2B P41595 1/20 0.37
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CDK1 P06493 1/20 0.37
CDK2 P24941 1/20 0.37
CDK9 P50750 1/20 0.37
GSK3B P49841 1/20 0.36
PDE2A O00408 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8576057 0.95 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL1552957 0.88 PDE4D (0.54) PDE4APDE4BPDE4CPDE4DPARP1
Hydrochloric Acid SCHEMBL8568573 0.87 PDE4D (0.53) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL1553709 0.87 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL1554160 0.84 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL1554161 0.82 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DPARP1
Hydrochloric Acid SCHEMBL8576071 0.82 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL1581071 0.81 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL1553706 0.80 PDE4D (0.71) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL8573500 0.80 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed