SCHEMBL8568827

SCHEMBL8568827

CC(=O)NCC(C)C(=O)N[C@@H](Cc1ccc(F)cc1)C(O)CN(CCC(C)C)C(=O)NC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 1/20 0.35
PSEN1 P49768 11/20 0.35
PSEN2 P49810 11/20 0.35
APH1B Q8WW43 11/20 0.35
NCSTN Q92542 11/20 0.35
APH1A Q96BI3 11/20 0.35
PSENEN Q9NZ42 11/20 0.35
BACE1 P56817 5/20 0.35
BACE2 Q9Y5Z0 2/20 0.34
CTSD P07339 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564050 0.91 CCR1 (0.35) TXNRD1PSEN1PSEN2APH1BNCSTN
SCHEMBL8984829 0.91 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5401511 0.87 CYP3A4 (0.37) TXNRD1PSEN1PSEN2APH1BNCSTN
SCHEMBL8569519 0.86 BACE1 (0.38) TXNRD1PSEN1PSEN2APH1BNCSTN
SCHEMBL8569492 0.84 PSEN1 (0.40) TXNRD1PSEN1PSEN2APH1BNCSTN
SCHEMBL8566334 0.83 PSEN1 (0.38) TXNRD1PSEN1PSEN2APH1BNCSTN
SCHEMBL8567291 0.82 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6443651 0.81 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6443658 0.81 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8568426 0.79 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558630-B1 RETROVIRAL PROTEASE INHIBITORS MONSANTO CO (US) 1998-04-08 EP claimed
US-5482947-A ENZYME INHIBITORS FOR HIV PROTEASE INHIBITION FROM UREA OR THIOUREA COMPOUNDS TALLEY JOHN J (US) 1996-01-09 US claimed