SCHEMBL8568869

SCHEMBL8568869

O=C1C(Cl)=C(N2CCCC2)C(=O)c2ccccc21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 6/20 0.73
TDP2 O95551 3/20 0.73
PLA2G1B P04054 1/20 0.73
ATG4B Q9Y4P1 1/20 0.73
MAPT P10636 10/20 0.63
APAF1 O14727 7/20 0.63
KMT2A Q03164 4/20 0.63
POLB P06746 3/20 0.63
HKDC1 Q2TB90 3/20 0.63
CASP3 P42574 2/20 0.63
GALK1 P51570 2/20 0.63
SENP8 Q96LD8 2/20 0.63
SENP7 Q9BQF6 2/20 0.63
SENP6 Q9GZR1 2/20 0.63
THRB P10828 1/20 0.63
RECQL P46063 1/20 0.63
SAE1 Q9UBE0 1/20 0.63
UBA2 Q9UBT2 1/20 0.63
ALDH1A1 P00352 9/20 0.61
L3MBTL1 Q9Y468 8/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10446114 0.98 NSD2 (0.71) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL17249910 0.86 NSD2 (0.88) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL17250437 0.86 NSD2 (0.60) NSD2TDP2PLA2G1BATG4BMAPT
2-Chloro-3-Morpholino-1,4-Naphthoquinone SCHEMBL29590404 0.84 NSD2 (0.67) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL8651868 0.84 NSD2 (1.00) NSD2TDP2PLA2G1BATG4BMAPT
2-Chloro-3-Morpholino-1,4-Naphthoquinone SCHEMBL197256 0.84 NSD2 (0.67) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL10556652 0.84 NSD2 (0.67) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL17249912 0.84 NSD2 (0.71) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL1242685 0.84 MAPT (0.67) NSD2TDP2PLA2G1BATG4BMAPT
SCHEMBL18266879 0.82 NSD2 (0.68) NSD2TDP2PLA2G1BATG4BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4324852-A REDOX COUPLES EASTMAN KODAK COMPANY (US) 1982-04-13 US claimed
US-4201588-A NONSILVER PHOTOGRAPHIC FILMS; DISULFIDE, DIAZOANTHRONE, DIAZOPHENANTHRONE, AROMATIC AZIDE, CARBAZIDES OR QUINONES AS PHOTOREDUCTANT; EXTERNAL HYDROGEN SOURCE EASTMAN KODAK COMPANY (US) 1980-05-06 US claimed
US-4195998-A NONSILVER PHOTOGRAPHIC FILMS; DISULFIDE, DIAZOANTHRONE, DIAZOPHENANTHRONE, AROMATIC AZIDE, QUINONE OR CARBAZIDE PHOTOREDUCTANT EASTMAN KODAK COMPANY (US) 1980-04-01 US claimed
US-5807898-A ASPIDIN, DESASPIDIN, METHYLENEBISASPIDINOL KAPADIA GOVIND J (US) 1998-09-15 US disclosed
US-5684035-A NAPHTHOQUINONES KAPADIA GOVIND J (US) 1997-11-04 US disclosed
US-4332884-A USING A DIOXIME CHELATING AGENT RICOH CO., LTD. (JP) 1982-06-01 US disclosed
US-4306014-A AMMONIA OR AMINES SUPPRESS THE COLOR-FORMING REACTION SYSTEM RICOH CO., LTD. (JP) 1981-12-15 US disclosed
US-4201588-A NONSILVER PHOTOGRAPHIC FILMS; DISULFIDE, DIAZOANTHRONE, DIAZOPHENANTHRONE, AROMATIC AZIDE, CARBAZIDES OR QUINONES AS PHOTOREDUCTANT; EXTERNAL HYDROGEN SOURCE EASTMAN KODAK COMPANY (US) 1980-05-06 US disclosed
US-4171221-A NONSILVER PHOTOGTAPHY EASTMAN KODAK COMPANY (US) 1979-10-16 US disclosed