SCHEMBL8569221

SCHEMBL8569221

COc1ccc2c(c1)[nH]c(=O)c1cccn12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.62
PARP1 P09874 13/20 0.59
MAP4K4 O95819 2/20 0.51
CSF1R P07333 2/20 0.51
MKNK2 Q9HBH9 2/20 0.51
DCLK1 O15075 1/20 0.51
PIM1 P11309 1/20 0.51
CSNK1D P48730 1/20 0.51
CDK5 Q00535 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
STK17A Q9UEE5 1/20 0.51
CDC7 O00311 1/20 0.48
PLK4 O00444 1/20 0.48
AURKA O14965 1/20 0.48
MAPK13 O15264 1/20 0.48
PDPK1 O15530 1/20 0.48
DYRK3 O43781 1/20 0.48
PRKD3 O94806 1/20 0.48
PAK4 O96013 1/20 0.48
ERBB2 P04626 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21755742 0.88 PARP1 (0.59) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL8564331 0.80 TP53 (0.68) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL13711927 0.80 TP53 (0.59) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL13711924 0.79 PARP1 (0.61) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL29893230 0.78 PARP1 (0.62) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL3339424 0.78 PARP1 (0.62) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL709373 0.78 PARP1 (0.47) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL4521450 0.78 TP53 (0.56) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL13082234 0.77 TP53 (0.68) TP53PARP1MAP4K4CSF1RMKNK2
SCHEMBL9415217 0.77 TP53 (0.68) TP53PARP1MAP4K4CSF1RMKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed