SCHEMBL8569394

SCHEMBL8569394

O=C(O)[C@H]1CC[C@H](Nc2ccc3ncnc(Nc4ccc(F)c(Cl)c4)c3n2)CC1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.61
ERBB2 P04626 8/20 0.61
HPGD P15428 1/20 0.54
HTT P42858 1/20 0.54
CSNK2A1 P68400 1/20 0.49
DYRK1A Q13627 1/20 0.46
HDAC3 O15379 2/20 0.45
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC10 Q969S8 2/20 0.45
HDAC11 Q96DB2 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569397 1.00 EGFR (0.61) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8570045 0.87 EGFR (0.59) EGFRERBB2HPGDHTTMAPT
SCHEMBL6993876 0.86 EGFR (0.72) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL6993885 0.86 EGFR (0.72) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8570632 0.84 EGFR (0.56) EGFRERBB2HPGDHTTDYRK1A
SCHEMBL6999421 0.82 EGFR (0.68) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8314168 0.79 EGFR (0.52) EGFRERBB2HPGDHTTMAPT
SCHEMBL8314173 0.79 EGFR (0.52) EGFRERBB2HPGDHTTMAPT
SCHEMBL8317027 0.78 EGFR (0.60) EGFRERBB2HPGDHTTCSNK2A1
SCHEMBL8317032 0.78 EGFR (0.60) EGFRERBB2HPGDHTTCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885226-A1 4-AMINO PYRIMIDINE DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997032881-A1 4-AMINO PYRIMIDINE DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1997-09-12 WO disclosed