SCHEMBL8570215

SCHEMBL8570215

COc1ccc(C(=O)Cl)c2[nH]c(-c3cccnc3)nc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.48
PKN1 Q16512 1/20 0.46
PKN2 Q16513 1/20 0.46
MKNK1 Q9BUB5 2/20 0.46
MKNK2 Q9HBH9 2/20 0.46
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
NPY5R Q15761 1/20 0.44
GSK3B P49841 2/20 0.42
DHODH Q02127 3/20 0.42
CYP11B1 P15538 3/20 0.42
CYP11B2 P19099 3/20 0.42
CYP17A1 P05093 2/20 0.42
CYP19A1 P11511 1/20 0.42
PARP1 P09874 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
HPSE Q9Y251 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP3A4 P08684 1/20 0.41
PNP P00491 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1554187 0.90 DHODH (0.50) NPC1PKN1PKN2MKNK1MKNK2
Hydrochloric Acid SCHEMBL8570223 0.89 DHODH (0.49) NPC1PKN1PKN2MKNK1MKNK2
SCHEMBL1553002 0.89 NPC1 (0.48) NPC1PKN1PKN2MKNK1MKNK2
SCHEMBL8653067 0.87 TNKS (0.51) GSK3BDHODHPARP1PARP2HPSE
SCHEMBL1553232 0.83 PDE4D (0.59)
SCHEMBL8603042 0.81 PDE4A (0.48) NPC1MKNK1MKNK2ALDH1A1DHODH
SCHEMBL8571233 0.80 NPC1 (0.46) NPC1PKN1PKN2MKNK1MKNK2
SCHEMBL4702865 0.78 NPC1 (0.72) NPC1MKNK1MKNK2ALDH1A1CYP11B1
SCHEMBL1553486 0.77 DHODH (0.57) ALDH1A1GSK3BDHODHPARP1PARP2
Hydrochloric Acid SCHEMBL8653073 0.76 DHODH (0.56) ALDH1A1GSK3BDHODHPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed