SCHEMBL8570672

SCHEMBL8570672

CNC(=O)c1c(O)c2ccccc2n(Cc2ccccc2)c1=O

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.74
HIF1A Q16665 1/20 0.68
KDM4E B2RXH2 3/20 0.66
GSK3B P49841 2/20 0.65
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
L3MBTL1 Q9Y468 2/20 0.62
HTT P42858 2/20 0.62
LMNA P02545 1/20 0.62
ALOX15 P16050 1/20 0.62
MAPK1 P28482 1/20 0.62
HSD17B10 Q99714 1/20 0.62
TDP1 Q9NUW8 1/20 0.60
POLB P06746 1/20 0.60
ALDH1A1 P00352 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18383362 0.85 EGLN1 (0.83) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL8244419 0.85 EGLN1 (1.00) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL5330412 0.83 EGLN1 (0.83) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL1440727 0.83 EGLN1 (0.67) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL19434051 0.81 HIF1A (0.77) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL24054656 0.80 HIF1A (0.72) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL16522300 0.80 GSK3B (0.79) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL24054539 0.80 MEN1 (0.72) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL24054669 0.80 MEN1 (0.74) EGLN1HIF1AKDM4EGSK3BMEN1
SCHEMBL1522936 0.80 KDM4E (0.81) EGLN1HIF1AKDM4EGSK3BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012066478-A1 QUINOLINONE DERIVATIVES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-05-24 WO disclosed