SCHEMBL8575587

SCHEMBL8575587

COc1ccccc1COc1nc2ccccc2c(-c2ccc3c(c2)OCO3)c1CC(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.51
KMT2A Q03164 6/20 0.51
MAPK1 P28482 4/20 0.51
HSD17B10 Q99714 4/20 0.51
CYP1A2 P05177 4/20 0.51
CYP3A4 P08684 4/20 0.51
CYP2D6 P10635 4/20 0.51
CYP2C19 P33261 4/20 0.51
LMNA P02545 3/20 0.51
CYP2C9 P11712 3/20 0.51
CLK4 Q9HAZ1 2/20 0.51
USP2 O75604 2/20 0.51
RECQL P46063 1/20 0.51
EDNRB P24530 6/20 0.51
ALDH1A1 P00352 3/20 0.47
TSHR P16473 3/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
TP53 P04637 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27461879 0.85 CYP1A2 (0.56) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL8577077 0.77 EDNRB (0.67) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL6314927 0.76 EDNRB (0.79) MAPK1EDNRBALDH1A1HPGDEDNRA
SCHEMBL8798051 0.76 EDNRB (0.57) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL8577921 0.76 EDNRB (0.61) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL8653767 0.76 EDNRB (0.52) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL8798547 0.75 EDNRB (0.56) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL8804966 0.71 EDNRB (0.58) MEN1KMT2AMAPK1HSD17B10CYP1A2
SCHEMBL8577086 0.69 TP53 (0.58) MEN1KMT2AMAPK1HSD17B10CYP1A2
Graveolinine SCHEMBL25286396 0.69 KDM4E (0.66) MEN1KMT2AMAPK1HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731321-A Endothelin receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-03-24 US disclosed