SCHEMBL8577283

SCHEMBL8577283

CCC(=O)NCc1cccc(Nc2n[nH]c3ncnc(Nc4cccc(Cl)c4)c23)c1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.68
CDK1 P06493 11/20 0.68
SRC P12931 9/20 0.68
ABL1 P00519 13/20 0.64
PRKCA P17252 11/20 0.64
PDGFRB P09619 3/20 0.49
PDGFRA P16234 3/20 0.49
ABL2 P42684 2/20 0.47
AURKA O14965 1/20 0.46
RPS6KB1 P23443 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577275 0.94 EGFR (0.63) EGFRCDK1SRCABL1PRKCA
SCHEMBL6186563 0.91 EGFR (0.70) EGFRCDK1SRCABL1PRKCA
SCHEMBL8125545 0.90 EGFR (0.71) EGFRCDK1SRCABL1PRKCA
SCHEMBL6184839 0.89 EGFR (0.72) EGFRCDK1SRCABL1PRKCA
SCHEMBL6190152 0.88 EGFR (0.65) EGFRCDK1SRCABL1PRKCA
SCHEMBL6191605 0.87 EGFR (0.66) EGFRCDK1SRCABL1PRKCA
SCHEMBL6189838 0.86 EGFR (0.64) EGFRCDK1SRCABL1PRKCA
SCHEMBL6186182 0.85 EGFR (0.64) EGFRCDK1SRCABL1PRKCA
SCHEMBL8581909 0.85 EGFR (0.60) EGFRCDK1SRCABL1PRKCA
SCHEMBL6185513 0.85 EGFR (0.59) EGFRCDK1SRCABL1PRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998014449-A1 FUSED PYRAZOLE DERIVATIVES AND PROCESSES FOR THEIR PREPARATION NOVARTIS AG (CH) 1998-04-09 WO claimed