SCHEMBL8577453

SCHEMBL8577453

CCCn1c(=O)c2[nH]c(C3CCCC3)nc2n(CCCc2ccc(OCC(=O)OC)cc2)c1=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 13/20 0.65
ADORA2A P29274 3/20 0.62
ADORA2B P29275 3/20 0.62
ADORA3 P0DMS8 2/20 0.60
GMNN O75496 2/20 0.60
LMNA P02545 2/20 0.60
TSHR P16473 2/20 0.60
PMP22 Q01453 2/20 0.60
HIF1A Q16665 2/20 0.60
MEN1 O00255 1/20 0.60
CYP1A2 P05177 1/20 0.60
KMT2A Q03164 1/20 0.60
NPC1 O15118 1/20 0.54
ALDH1A1 P00352 1/20 0.54
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
NFKB1 P19838 1/20 0.54
MAPK1 P28482 1/20 0.54
RAB9A P51151 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8576785 0.93 ADORA1 (0.64) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8580875 0.92 ADORA1 (0.67) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8578133 0.91 ADORA1 (0.66) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8579411 0.88 ADORA1 (0.73) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8579611 0.88 ADORA1 (0.68) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8578025 0.87 ADORA1 (0.65) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8577917 0.87 ADORA1 (0.69) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8577863 0.85 ADORA1 (0.55) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8579158 0.84 ADORA1 (0.76) ADORA1ADORA2AADORA2BADORA3GMNN
SCHEMBL8576983 0.83 ADORA2A (0.79) ADORA1ADORA2AADORA2BADORA3GMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed