SCHEMBL8580401

SCHEMBL8580401

CC=C[C@H]1COc2ccc(C(=O)NN(C(=O)c3cc(C)cc(C)c3)C(C)(C)C)c(C)c2O1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 7/20 0.49
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8594670 0.91 ABCB1 (0.51) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL3766544 0.91 ABCB1 (0.51) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL14078518 0.90 ABCB1 (0.50) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL3771854 0.88 ABCB1 (0.48) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL16368762 0.88 ABCB1 (0.48) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL13003212 0.88 ABCB1 (0.48) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL13060027 0.88 ABCB1 (0.48) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL3769756 0.85 ABCB1 (0.51) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL8617673 0.85 ABCB1 (0.51) ABCB1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL13003215 0.84 ABCB1 (0.51) ABCB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2455375-A2 Diacylhydrazine ligands for modulating the expression of exogenous genes in mammalian systems via an ecdysone receptor complex Intrexon Corporation (US) 2012-05-23 EP disclosed