SCHEMBL8582252

SCHEMBL8582252

CC(=O)N[C@H](CC(=O)OC(C)(C)C)C(=O)S

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.43
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
NFKB1 P19838 1/20 0.39
PTGS2 P35354 1/20 0.39
THPO P40225 1/20 0.39
RECQL P46063 1/20 0.39
BLM P54132 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ALDH1A1 P00352 1/20 0.34
CTSK P43235 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577814 0.86 CYP2D6 (0.54) CYP2D6SMN1; SMN2HDAC1HDAC6CTSK
SCHEMBL11912121 0.84 MAPT (0.48) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL31023862 0.84 CYP2D6 (0.44) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL31023961 0.84 CYP2D6 (0.44) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL13259810 0.84 MAPT (0.48) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL25192292 0.84 MAPT (0.48) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL8582254 0.81 CYP2D6 (0.42) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL13033062 0.81 CYP2D6 (0.45) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL16945945 0.79 GNPAT (0.47) CYP2D6KDM4EMAPTTHRBALOX15
SCHEMBL16945887 0.79 GNPAT (0.47) CYP2D6KDM4EMAPTTHRBALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705527-A VASODILATORS AND ANGINA PECTORIS SANKYO COMPANY, LIMITED (JP) 1998-01-06 US disclosed
EP-0641769-B1 AMINO ACID DERIVATIVE SANKYO CO (JP) 1997-01-29 EP disclosed
EP-0641769-A1 AMINO ACID DERIVATIVE SANKYO COMPANY LIMITED (JP) 1995-03-08 EP disclosed