SCHEMBL8583142

SCHEMBL8583142

COC(=O)C(C)(C(=O)C(C)(C(=O)OC)c1ccccc1)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.62
NPSR1 Q6W5P4 1/20 0.47
SRC P12931 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
KMT2A Q03164 3/20 0.44
MAPT P10636 2/20 0.44
CES1 P23141 1/20 0.43
ELANE P08246 1/20 0.42
CYP2C19 P33261 2/20 0.42
HIF1A Q16665 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16732028 0.92 KCNN4 (0.67) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL1561399 0.88 KCNN4 (0.62) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL8784152 0.88 KCNN4 (0.62) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL28932488 0.86 KCNN4 (0.60) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL1561571 0.85 KCNN4 (0.58) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL9383813 0.85 KCNN4 (0.58) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL728471 0.79 KCNN4 (0.67) KCNN4NPSR1SRCHDAC3HDAC4
SCHEMBL4022191 0.79 KCNN4 (0.67) KCNN4SRCHDAC3HDAC4HDAC1
SCHEMBL28778735 0.78 KCNN4 (0.42) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL1682976 0.78 KCNN4 (0.64) KCNN4NPSR1SRCHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840614-A1 CALPAIN INHIBITORS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SANOFI WINTHROP, INC. (US) 1998-05-13 EP disclosed
WO-1996041638-A1 CALPAIN INHIBITORS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SANOFI WINTHROP, INC. (US) 1996-12-27 WO disclosed