SCHEMBL858440

SCHEMBL858440

COC(C)C(c1nc2cc(I)ccc2[nH]1)N1C(=O)NC(c2ccc(OCCO)cc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 2/20 0.39
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
P2RY12 Q9H244 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
CHEK2 O96017 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13950575 1.00 MAP2K1 (0.39) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL844242 1.00 MAP2K1 (0.39) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL843942 1.00 MAP2K1 (0.39) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL843963 0.93 MAP2K1 (0.41) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL13950768 0.93 MAP2K1 (0.41) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL843962 0.93 MAP2K1 (0.41) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL13765313 0.88 MAP2K1 (0.49) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL10076794 0.88 MAP2K1 (0.49) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL4023862 0.86 MAP2K1 (0.38) MAP2K1PDE3BPDE3AP2RY12ESR1
SCHEMBL859794 0.84 MAP2K1 (0.37) MAP2K1PDE3BPDE3AP2RY12ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188276-B1 SUBSTITUTED HYDANTOINS HOFFMANN LA ROCHE (CH) 2012-03-28 EP disclosed