SCHEMBL8601328

SCHEMBL8601328

O=Cc1c2ccccc2cc2ccc(Cl)cc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.49
CYP2A6 P11509 1/20 0.45
MAPT P10636 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
AHR P35869 1/20 0.40
L3MBTL1 Q9Y468 4/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 3/20 0.39
GAA P10253 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HIF1A Q16665 1/20 0.38
CYP1B1 Q16678 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488182 0.89 CYP2A6 (0.45) ERN1CYP2A6MAPTCYP1A2CYP2C9
SCHEMBL29388184 0.84 ERN1 (0.57) ERN1CYP2A6MAPTCYP1A2CYP2C9
SCHEMBL342278 0.84 ERN1 (0.57) ERN1CYP2A6MAPTCYP1A2CYP2C9
SCHEMBL10997990 0.81 SLC2A1 (0.46) ERN1CYP2A6MAPTAHRSMN1; SMN2
SCHEMBL4893713 0.81 ERN1 (0.50) ERN1CYP2A6MAPTCYP1A2CYP2C9
SCHEMBL14643530 0.80 ERN1 (0.47) ERN1CYP2A6MAPTCYP1A2CYP2C9
Hydrochloric Acid SCHEMBL11307480 0.79 SLC2A1 (0.49) ERN1CYP2A6MAPTAHRSMN1; SMN2
SCHEMBL19960402 0.79 ERN1 (0.46) ERN1CYP2A6MAPTCYP1A2CYP2C9
Methyl Alcohol SCHEMBL27670101 0.79 ERN1 (0.57) ERN1CYP2A6MAPTCYP1A2CYP2C9
SCHEMBL5748504 0.79 ERN1 (0.49) ERN1MAPTCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719166-A TREATING PSYCHOSES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1998-02-17 US disclosed
US-5681840-A ANTIDOPAMINERGIC AGENTS ZENECA LIMITED (GB) 1997-10-28 US disclosed
EP-0532178-B1 Methanoanthracenes as dopamine antagonists ZENECA LTD (GB) 1996-10-16 EP disclosed
EP-0533344-B1 Methanoanthracenes as dopamine antagonists ZENECA LTD (GB) 1996-10-16 EP disclosed
EP-0532177-B1 Methanoanthracenes as dopamine antagonists ZENECA LTD (GB) 1996-10-16 EP disclosed
US-5550136-A ANTAGONISTS OF DOPAMINE D-2 RECEPTORS ZENECA LIMITED (GB) 1996-08-27 US disclosed
US-5512575-A ANTISEROTONINE AGENT ZENECA LIMITED (GB) 1996-04-30 US disclosed
US-5455246-A Treating neuropsychiatric disorders IMPERIAL CHEMICAL INDUSTRIES, PLC (GB) 1995-10-03 US disclosed
US-5399568-A Dopamine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-03-21 US disclosed
US-5266570-A Neuropsychiatric disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-11-30 US disclosed
US-4803226-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4803221-A Anthracene derivatives BURROUGHS WELLCOME CO. (US) 1989-02-07 US disclosed
US-4719047-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP disclosed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed
US-4340624-A STYRYL-LIKE COMPOUNDS MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 1982-07-20 US disclosed
US-4088772-A TRANQUILIZERS, ANALGESICS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-05-09 US disclosed
US-4077977-A Ethenoanthracenes E. I. DU PONT DE NEMOURS AND COMPANY (US) 1978-03-07 US disclosed
US-4017313-A Photosensitive composition containing a leuco dye, a photosensitizer, an aromatic aldehyde and a secondary or tertiary amine and the use thereof in a direct-print process E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-04-12 US disclosed