SCHEMBL8607133

SCHEMBL8607133

OCc1cc(-c2cccc(C(F)(F)F)c2)no1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.62
P2RY14 Q15391 3/20 0.49
TSPO P30536 2/20 0.47
CYP2C9 P11712 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
HTT P42858 1/20 0.47
ALDH1A1 P00352 1/20 0.46
HRH1 P35367 1/20 0.46
OPRD1 P41143 1/20 0.46
MAOB P27338 2/20 0.46
IDO1 P14902 1/20 0.46
BRD4 O60885 1/20 0.45
S1PR1 P21453 1/20 0.45
KMO O15229 2/20 0.44
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1221497 0.85 NOTUM (0.48) NOTUMCYP2C9NPC1RAB9AHTT
SCHEMBL11397855 0.85 NPC1 (0.47) NOTUMCYP2C9NPC1RAB9AHTT
SCHEMBL1441397 0.84 NOTUM (0.56) NOTUMP2RY14TSPOCYP2C9TMEM97
SCHEMBL2120020 0.83 NOTUM (0.64) NOTUMP2RY14TSPOCYP2C9TMEM97
SCHEMBL12017168 0.78 NOTUM (0.49) NOTUMP2RY14TSPOCYP2C9TMEM97
SCHEMBL1313626 0.77 NOTUM (1.00) NOTUMCYP2C9NPC1RAB9AHTT
SCHEMBL1544352 0.77 NOTUM (0.72) NOTUMCYP2C9NPC1RAB9A
SCHEMBL2318106 0.77 KDR (0.60) NOTUMNPC1RAB9AHTTALDH1A1
SCHEMBL23221331 0.75 NPC1 (0.51) NOTUMNPC1RAB9AHTTALDH1A1
SCHEMBL1198267 0.74 KDM4E (0.59) SIGMAR1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998015541-A1 NOVEL ISOXAZOL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS Gyógyszergyár Rt. (HU) 1998-04-16 WO disclosed