SCHEMBL8613151

SCHEMBL8613151

CN(C)c1ncnc2c1ncn2[C@@H]1O[C@H](COC(c2ccccc2)(c2ccccc2)c2ccccc2)[C@@H](O)[C@H]1OC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TYMP P19971 11/20 0.63
ADORA1 P30542 2/20 0.54
ANPEP P15144 3/20 0.49
NPEPPS P55786 3/20 0.49
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8610268 0.93 TYMP (0.63) TYMPADORA1ANPEPNPEPPSADORA2A
SCHEMBL8612735 0.88 TYMP (0.54) TYMPADORA1ANPEPNPEPPS
SCHEMBL8612740 0.88 TYMP (0.54) TYMPADORA1ANPEPNPEPPS
SCHEMBL8611837 0.88 TYMP (0.67) TYMPADORA1
SCHEMBL8612918 0.87 TYMP (0.52) TYMPADORA1
SCHEMBL8613000 0.87 TYMP (0.83) TYMPADORA1
SCHEMBL8612341 0.86 TYMP (0.63) TYMPADORA1
SCHEMBL8614133 0.85 TYMP (0.64) TYMPADORA1
SCHEMBL18797886 0.84 TYMP (0.62) TYMPADORA1
SCHEMBL31160244 0.84 TYMP (0.62) TYMPADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO claimed
US-5750675-A 2'-\"up\" fluorinated 2'-deoxy-arabinofuranosylpurines SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1998-05-12 US disclosed
US-5525720-A Synthesis of 2'-\"up\" fluorinated 2'-deoxy-arabinofuranosyl purines SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1996-06-11 US disclosed
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO disclosed