SCHEMBL8615959

SCHEMBL8615959

NC1=N[C@@]2(CO1)c1cc(-c3cncnc3)ccc1O[C@H]1CCC(=O)CC12

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.70
CTSD P07339 4/20 0.70
CYP2D6 P10635 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9932000 1.00 BACE1 (0.70) BACE1CTSDCYP2D6
SCHEMBL9931666 0.89 BACE1 (0.72) BACE1CTSDCYP2D6
SCHEMBL9931668 0.89 BACE1 (0.72) BACE1CTSDCYP2D6
SCHEMBL9931773 0.89 BACE1 (0.70) BACE1CTSDCYP2D6
SCHEMBL9931420 0.87 BACE1 (0.57) BACE1CTSDCYP2D6
SCHEMBL9931422 0.87 BACE1 (0.57) BACE1CTSDCYP2D6
SCHEMBL9932306 0.85 BACE1 (0.77) BACE1CTSDCYP2D6
SCHEMBL9882484 0.85 BACE1 (0.77) BACE1CTSDCYP2D6
SCHEMBL10237838 0.85 BACE1 (0.77) BACE1CTSDCYP2D6
SCHEMBL9931493 0.84 BACE1 (0.57) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071458-A1 HETEROCYCLIC INHIBITORS OF BETA - SECRETASE FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2012-05-31 WO disclosed