SCHEMBL8617907

SCHEMBL8617907

[CH2]CC#Cc1cccc(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.56
CHRM1 P11229 3/20 0.56
CHRM3 P20309 3/20 0.56
GRM5 P41594 5/20 0.50
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA9 Q16790 2/20 0.50
FFAR1 O14842 1/20 0.48
CHRM4 P08173 2/20 0.43
CHRM5 P08912 2/20 0.43
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23843579 0.84 CHRM2 (0.57) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL30707880 0.82 GRM5 (0.66) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL6132140 0.82 GRM5 (0.66) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL2155272 0.82 CHRM2 (0.56) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL19291472 0.82 CHRM2 (0.56) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL29745229 0.82 CHRM2 (0.56) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL5886631 0.81 CHRM2 (0.52) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL7601866 0.81 GRM5 (0.56) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL29994376 0.81 GRM5 (0.56) CHRM2CHRM1CHRM3GRM5CA12
SCHEMBL16298669 0.81 CHRM2 (0.55) CHRM2CHRM1CHRM3GRM5CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5733914-A Pyrido 2, 3-d!pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation WARNER-LAMBERT COMPANY (US) 1998-03-31 US disclosed
US-5620981-A ANTICARCINOGENIC AGENTS, ATHEROSCLEROSIS, RESTENOSIS, PSORIASIS WARNER-LAMBERT COMPANY (US) 1997-04-15 US disclosed