SCHEMBL8619916

SCHEMBL8619916

COc1c(N2CC[C@@H](C(N)CF)C2)c(F)c(N)c2c(=O)c(C(=O)O)cn([C@@H]3C[C@@H]3F)c12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.50
CYP3A4 P08684 1/20 0.45
POLB P06746 2/20 0.44
CACNA1F O60840 1/20 0.44
MAPK1 P28482 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
GSK3B P49841 6/20 0.43
SLC2A1 P11166 1/20 0.40
KDM4E B2RXH2 1/20 0.39
PRKD3 O94806 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
OPRM1 P35372 1/20 0.39
CLK2 P49760 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6163513 0.82 CYP3A4 (0.50) KCNH2CYP3A4POLBCACNA1FMAPK1
SCHEMBL7463545 0.82 KCNH2 (0.48) KCNH2CYP3A4POLBCACNA1FMAPK1
SCHEMBL7468912 0.82 KCNH2 (0.48) KCNH2CYP3A4POLBCACNA1FMAPK1
SCHEMBL8324629 0.82 KCNH2 (0.72) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL8332205 0.82 KCNH2 (0.72) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL8331341 0.82 KCNH2 (0.72) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL6959217 0.81 KCNH2 (0.58) KCNH2CYP3A4POLBCACNA1FMAPK1
SCHEMBL5619269 0.81 KCNH2 (0.58) KCNH2CYP3A4POLBCACNA1FMAPK1
SCHEMBL5619262 0.81 KCNH2 (0.58) KCNH2CYP3A4POLBCACNA1FMAPK1
SCHEMBL8544340 0.81 KCNH2 (0.58) KCNH2CYP3A4POLBCACNA1FMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10287669-A None JP disclosed
JP-H10287669-A SUBSTITUTED AMINOMETHYLPYRROLIDINE DERIVATIVE DAI ICHI SEIYAKU CO LTD 1998-10-27 JP disclosed