SCHEMBL8620143

SCHEMBL8620143

COc1ccc(Cc2nc3c(C(N)=O)cccc3[nH]2)cc1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.65
PLA2G2A P14555 1/20 0.65
ALOX15 P16050 1/20 0.65
PTGS2 P35354 1/20 0.65
CD38 P28907 1/20 0.52
GRIN1 Q05586 1/20 0.51
GRIN2B Q13224 1/20 0.51
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
CHEK2 O96017 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6841346 0.83 PARP1 (0.61) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL6842032 0.82 PARP1 (0.60) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL10869434 0.81 GRIN1 (0.74) GRIN1GRIN2B
SCHEMBL6842016 0.81 PARP1 (0.61) PARP1PLA2G2AALOX15PTGS2HDAC3
Hydrochloric Acid SCHEMBL10410762 0.80 GRIN1 (0.73) GRIN1GRIN2B
SCHEMBL23581718 0.80 PARP1 (0.61) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL7319077 0.79 PARP1 (1.00) PARP1PLA2G2AALOX15PTGS2CHEK2
Hydrochloric Acid SCHEMBL28060188 0.79 PARP1 (0.59) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL23581692 0.78 PARP1 (0.66) PARP1CHEK2
SCHEMBL25022851 0.76 PARP1 (0.63) PARP1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841924-A1 BENZIMIDAZOLE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1998-05-20 EP disclosed
WO-1997004771-A1 BENZIMIDAZOLE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1997-02-13 WO disclosed