SCHEMBL8620522

SCHEMBL8620522

Nc1nc(N)c2ncn(CC(CF)OCP)c2n1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 3/20 0.51
CDK2 P24941 3/20 0.51
CDK1 P06493 2/20 0.51
CCNB1 P14635 2/20 0.51
HPRT1 P00492 6/20 0.45
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
SLC29A1 Q99808 1/20 0.39
ADORA2A P29274 2/20 0.36
ADORA1 P30542 1/20 0.36
AHCY P23526 2/20 0.36
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3860366 1.00 CCNE1 (0.51) CCNE1CDK2CDK1CCNB1HPRT1
SCHEMBL465830 0.88 CCNE1 (0.51) CCNE1CDK2CDK1CCNB1HPRT1
SCHEMBL384146 0.84 ADORA2A (0.54) ADORA2AADORA1AHCY
SCHEMBL6366274 0.84 ADORA2A (0.54) ADORA2AADORA1AHCY
SCHEMBL29624179 0.82 HPRT1 (0.56) CCNE1CDK2CDK1CCNB1HPRT1
SCHEMBL9189595 0.82 CCNE1 (0.49) CCNE1CDK2CDK1CCNB1HPRT1
SCHEMBL3860363 0.82 HPRT1 (0.56) CCNE1CDK2CDK1CCNB1HPRT1
SCHEMBL9193126 0.82 HPRT1 (0.56) CCNE1CDK2CDK1CCNB1HPRT1
SCHEMBL3857976 0.82 CCNE1 (0.57) CCNE1CDK2CDK1CCNB1HSP90AA1
SCHEMBL3856997 0.79 HPRT1 (0.71) HPRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533833-B1 PHOSPHOROUS PRODUGS GLAZIER ARNOLD (US) 1995-12-20 EP claimed
US-5733896-A VIRICIDE FOR RETROVIRUS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1998-03-31 US disclosed
EP-0454427-B1 Antiretroviral bases ACAD OF SCIENCE CZECH REPUBLIC (CZ) 1995-12-06 EP disclosed
EP-0454427-A1 Antiretroviral bases Institute of Organic Chemistry and Biochemistry of the Academy of Sciences of the Czech Republic (CZ) 1991-10-30 EP disclosed