SCHEMBL8624640

SCHEMBL8624640

COC(=O)c1cccc2[nH]c(-c3cccc(C(F)(F)F)c3)nc12

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.73
PKN1 Q16512 2/20 0.64
PKN2 Q16513 2/20 0.64
DHODH Q02127 3/20 0.53
PIN1 Q13526 1/20 0.52
PLA2G2A P14555 1/20 0.48
ALOX15 P16050 1/20 0.48
PTGS2 P35354 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313257 0.88 PKN1 (0.74) PARP1PKN1PKN2DHODHPLA2G2A
SCHEMBL1891860 0.86 PARP1 (0.80) PARP1DHODHPIN1
Acetic Acid SCHEMBL7316877 0.85 PKN1 (0.69) PARP1PKN1PKN2DHODHPLA2G2A
SCHEMBL7317874 0.85 PARP1 (1.00) PARP1PKN1PKN2DHODH
SCHEMBL7322715 0.83 PKN1 (0.81) PARP1PKN1PKN2DHODHPLA2G2A
SCHEMBL1170810 0.81 PKN1 (0.77) PARP1PKN1PKN2DHODHPLA2G2A
SCHEMBL12673092 0.81 PARP1 (0.66) PARP1PKN1PKN2DHODHPIN1
SCHEMBL505325 0.81 PKN1 (0.77) PARP1PKN1PKN2DHODHPLA2G2A
SCHEMBL12673126 0.81 PARP1 (0.68) PARP1PKN1PKN2DHODHPIN1
SCHEMBL12673377 0.80 PARP1 (0.67) PARP1PKN1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841924-A1 BENZIMIDAZOLE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1998-05-20 EP disclosed
WO-1997004771-A1 BENZIMIDAZOLE COMPOUNDS NEWCASTLE UNIVERSITY VENTURES LIMITED (GB) 1997-02-13 WO disclosed