SCHEMBL8625264

SCHEMBL8625264

Cc1c(F)c(N2CCC(N)C2)cc2c1c(=O)c(C(=O)O)cn2-c1ccc(F)cc1F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.60
KCNH2 Q12809 1/20 0.51
HRH3 Q9Y5N1 1/20 0.51
TOP1 P11387 3/20 0.47
GSK3B P49841 2/20 0.47
EPHA2 P29317 1/20 0.47
FLT4 P35916 1/20 0.47
RARB P10826 1/20 0.47
TBXAS1 P24557 1/20 0.47
SLC6A3 Q01959 1/20 0.47
DYRK1A Q13627 2/20 0.47
PIM3 Q86V86 2/20 0.47
RPS6KB1 P23443 1/20 0.47
MATK P42679 1/20 0.47
MAPKAPK3 Q16644 1/20 0.47
AURKB Q96GD4 1/20 0.47
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8112209 0.99 KMT2A (0.59) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL5868715 0.95 KMT2A (0.55) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL8925800 0.89 KCNH2 (0.49) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL8924265 0.89 KCNH2 (0.49) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL8923585 0.89 KCNH2 (0.49) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL8923571 0.89 KCNH2 (0.49) KMT2AKCNH2HRH3TOP1GSK3B
Hydrochloric Acid SCHEMBL8110971 0.89 KCNH2 (0.51) KMT2AKCNH2HRH3TOP1DYRK1A
SCHEMBL8565238 0.88 KCNH2 (0.48) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL8565232 0.88 KCNH2 (0.48) KMT2AKCNH2HRH3TOP1GSK3B
SCHEMBL8564911 0.88 KCNH2 (0.48) KMT2AKCNH2HRH3TOP1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2815119-B2 1998-10-27 JP claimed
US-5563138-A 4-OXOQUINOLINE-3-CARBOXYLIC ACID COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1996-10-08 US claimed
EP-0398967-A1 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1990-11-28 EP claimed
EP-0326891-A2 Antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-08-09 EP claimed
WO-1989006649-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1989-07-27 WO claimed
US-5585491-A Antibacterial agents OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-12-17 US disclosed
EP-0398967-A1 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1990-11-28 EP disclosed
US-4920120-A 3-CARBOXY, 4-OXO, 6-FLUORO, 7-NITROGEN-CONTAINING RING 1,4-DIHYDRO-1,8-NAPHTHYRIDINES WARNER-LAMBERT COMPANY (US) 1990-04-24 US disclosed
EP-0326891-A2 Antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-08-09 EP disclosed
WO-1989006649-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1989-07-27 WO disclosed