SCHEMBL8625409

SCHEMBL8625409

CCOP(C)(=O)CS(=O)(=O)O

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
TP53 P04637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PPARD Q03181 2/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17445781 0.79 TSHR (0.42) TSHRTP53TDP1PPARDCA1
SCHEMBL2855157 0.79 TSHR (0.50) TSHRTP53TDP1PPARDCA12
SCHEMBL14141773 0.78 PPARD (0.39) TSHRTP53TDP1PPARDCA12
SCHEMBL8714812 0.77 TSHR (0.48) TSHRTP53TDP1PPARDCA12
SCHEMBL8623480 0.72 TSHR (0.36) TSHRTP53TDP1PPARDCA12
Diethyl Hydrogen Phosphate SCHEMBL19812734 0.71 TSHR (0.43) TSHRTP53TDP1PPARDCA12
SCHEMBL22829580 0.71 TSHR (0.39) TSHRTP53TDP1PPARDCA12
SCHEMBL8764678 0.70
Triethyl Phosphate SCHEMBL27295346 0.70 TSHR (0.72) TSHRTP53TDP1PPARDCA12
SCHEMBL22829573 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712396-A PHOSPHONOSULFONATE COMPOUNDS USED FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND ATHEROSCLEROSIS MAGNIN DAVID R (US) 1998-01-27 US disclosed
US-5567841-A ANTICHOLESTEROL AGENT BRISTOL-MYERS SQUIBB COMPANY (US) 1996-10-22 US disclosed
US-5470845-A Methods of using α-phosphonosulfonate squalene synthetase inhibitors including the treatment of atherosclerosis and hypercholesterolemia BRISTOL-MYERS SQUIBB COMPANY (US) 1995-11-28 US disclosed