SCHEMBL8627693

SCHEMBL8627693

CCOC(=O)C(c1ccc2c(c1)OCO2)C(C=O)c1ccc(OC)cc1OCC(=O)O.COc1ccc(C2(O)OC(=O)C(c3ccc4c(c3)OCO4)=C2Cc2ccc3nsnc3c2)c(OCC(=O)O)c1

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 20/20 0.52
EDNRB P24530 14/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829632 0.88 EDNRA (0.67) EDNRAEDNRB
SCHEMBL7842088 0.82 EDNRA (0.64) EDNRAEDNRB
SCHEMBL7839624 0.78 KMT2A (0.48) EDNRAEDNRB
SCHEMBL8037809 0.77 EDNRA (0.86) EDNRAEDNRB
SCHEMBL7840661 0.76 EDNRA (0.64) EDNRAEDNRB
SCHEMBL7842077 0.75 EDNRA (0.62) EDNRAEDNRB
SCHEMBL8147810 0.75 EDNRA (0.75) EDNRAEDNRB
SCHEMBL7839726 0.74 EDNRA (0.81) EDNRAEDNRB
SCHEMBL7841623 0.72 KMT2A (0.44) EDNRA
SCHEMBL7842300 0.72 EDNRA (0.57) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882030-A1 2,1,3-BENZOTHIA(OXA)DIAZOLE DERIVATIVES HAVING AN ENDOTHELIN RECEPTOR ANTAGONISTIC EFFECT MERCK PATENT GmbH (DE) 1998-12-09 EP disclosed
WO-1997030982-A1 2,1,3-BENZOTHIA(OXA)DIAZOLE DERIVATIVES HAVING AN ENDOTHELIN RECEPTOR ANTAGONISTIC EFFECT MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-08-28 WO disclosed