SCHEMBL8629442

SCHEMBL8629442

CC(c1cccnc1)c1scc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.43
HRH1 P35367 3/20 0.43
CHRM1 P11229 2/20 0.43
KCNH2 Q12809 2/20 0.43
CYP3A4 P08684 1/20 0.43
CFTR P13569 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
GOPC Q9HD26 1/20 0.42
KDM4E B2RXH2 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
KCNA5 P22460 2/20 0.39
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
TBXAS1 P24557 2/20 0.37
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 1/20 0.37
KCNN4 O15554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8597805 0.83 CYP3A4 (0.40) CYP2D6HRH1CHRM1KCNH2CYP3A4
SCHEMBL10446411 0.74 CFTR (0.58) CYP3A4CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL14283944 0.73 CFTR (0.63) KCNH2CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL17069338 0.73 CFTR (0.63) KCNH2CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL17071838 0.73 CFTR (0.63) KCNH2CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL2601115 0.73 CFTR (0.63) KCNH2CFTRSLC6A2SLC6A4SLC6A3
Ammonia Solution, Strong SCHEMBL5999497 0.71 CFTR (0.61) KCNH2CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL15780702 0.70 CCR4 (0.40) CYP3A4KDM4EGAATSHR
Ammonia Solution, Strong SCHEMBL354291 0.69 CCR4 (0.39) CYP3A4KDM4EGAATSHR
SCHEMBL6999631 0.68 TSHR (0.66) CYP2D6HRH1CHRM1KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed