SCHEMBL8630756

SCHEMBL8630756

COc1cc(C(=O)N2CCCC(CC(=O)N3CCCCC3)c3cc(F)ccc32)ccc1NC(=O)c1ccccc1C

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 10/20 0.46
AVPR1B P47901 5/20 0.46
AVPR2 P30518 10/20 0.45
ABCB11 O95342 1/20 0.43
HTR1A P08908 1/20 0.43
CHRM1 P11229 1/20 0.43
OXTR P30559 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRM1 P35372 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4681827 0.87 AVPR2 (0.60) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL7336268 0.87 AVPR2 (0.50) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL7334156 0.86 AVPR2 (0.51) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL7356805 0.85 AVPR1A (0.50) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL7353295 0.84 AVPR1A (0.49) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL7353413 0.84 AVPR1A (0.61) AVPR1AAVPR1BAVPR2ABCB11HTR1A
Hydrochloric Acid SCHEMBL7354302 0.81 AVPR1A (0.47) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL7353320 0.81 AVPR2 (0.55) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL4684981 0.81 AVPR2 (0.52) AVPR1AAVPR1BAVPR2ABCB11HTR1A
SCHEMBL4685964 0.80 AVPR2 (0.47) AVPR1AAVPR1BAVPR2ABCB11HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed