SCHEMBL863338

SCHEMBL863338

O=C1CCC(=O)N1c1cc(Cc2n[nH]c(=O)c3ccccc23)ccc1F

nearest known ligand 0.92

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.92
LMNA P02545 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29408705 1.00 PARP1 (0.92) PARP1LMNA
SCHEMBL3388183 0.96 PARP1 (1.00) PARP1
SCHEMBL3385144 0.91 PARP1 (0.80) PARP1LMNA
SCHEMBL3388610 0.89 PARP1 (1.00) PARP1
SCHEMBL3385663 0.87 PARP1 (0.77) PARP1LMNA
SCHEMBL13007107 0.86 PARP1 (0.70) PARP1LMNA
SCHEMBL30132754 0.86 PARP1 (0.73) PARP1LMNA
SCHEMBL25890317 0.86 PARP1 (0.73) PARP1LMNA
SCHEMBL4440678 0.86 PARP1 (0.79) PARP1
SCHEMBL13007009 0.86 PARP1 (0.72) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210244706-A1 DNA Damage Repair Inhibitors for Treatment of Cancer THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2021-08-12 US disclosed
US-20200155521-A1 PHARMACEUTICAL COMBINATION FOR TREATMENT OF CANCER ARQULE, INC. 2020-05-21 US disclosed
US-20170319543-A1 DNA DAMAGE REPAIR INHIBITORS FOR TREATMENT OF CANCER THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2017-11-09 US disclosed
EP-2305221-B1 DNA damage repair inhibitors for treatment of cancer KUDOS PHARM LTD (GB) 2015-05-20 EP disclosed
US-8143241-B2 DNA damage repair inhibitors for treatment of cancer KUDOS PHARMACEUTICALS LIMITED (GB) 2012-03-27 US disclosed
EP-2305221-A1 Dna damage repair inhibitors for treatment of cancer Kudos Pharmaceuticals Limited (GB) 2011-04-06 EP disclosed
EP-1501822-B1 PHTHALAZINONE DERIVATIVES KUDOS PHARM LTD (GB) 2010-12-15 EP disclosed
US-7196085-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2007-03-27 US disclosed
US-7196085-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2007-03-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170319543-A1 DNA DAMAGE REPAIR INHIBITORS FOR TREATMENT OF CANCER PARP2, MRE11, PARP1 PARP1 3/4885LMNA 1800/4885
US-20200155521-A1 PHARMACEUTICAL COMBINATION FOR TREATMENT OF CANCER TP53, KRAS, VHL PARP1 1298/4885LMNA 2164/4885
US-20210244706-A1 DNA Damage Repair Inhibitors for Treatment of Cancer PARP2, MRE11, PARP1 PARP1 3/4885LMNA 1800/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.