SCHEMBL8633754

SCHEMBL8633754

CC(C)N1C(=S)CC(C)(C)c2ccc(C#Cc3ccc(C(=O)O)cc3)cc21

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RARB P10826 20/20 0.80
RARG P13631 20/20 0.80
RARA P10276 17/20 0.80
CYP26A1 O43174 1/20 0.54
CYP3A4 P08684 1/20 0.54
CRABP2 P29373 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30590593 0.78 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8633422 0.78 RARB (0.61) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8604441 0.78 RARB (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8633755 0.76 RARB (0.66) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8634937 0.75 RARB (0.74) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8866606 0.74 RARB (0.76) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6577982 0.73 RARB (0.66) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8631779 0.71 RARB (0.65) RARBRARGRARACYP26A1CYP3A4
SCHEMBL17675629 0.71 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL31725168 0.71 RARB (1.00) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825986-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1998-03-04 EP claimed
WO-1996036609-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-11-21 WO claimed