SCHEMBL8640738

SCHEMBL8640738

O=C(c1ccccc1)N1CC[C@](CCO)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 17/20 0.67
TACR1 P25103 15/20 0.67
TACR3 P29371 6/20 0.58
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HRH1 P35367 1/20 0.53
CCR5 P51681 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954575 1.00 TACR2 (0.67) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6950742 0.93 TACR2 (0.66) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL8810221 0.91 TACR2 (0.56) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL8119487 0.87 EPHX2 (0.57) TACR2TACR1TACR3CYP2D6CCR5
SCHEMBL7132390 0.87 TACR2 (0.69) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6544551 0.87 TACR2 (0.69) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL6998425 0.86 EPHX2 (0.53) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL7958373 0.86 TACR2 (0.52) TACR2TACR1TACR3CYP3A4CYP2D6
SCHEMBL8640624 0.86 TACR2 (0.52) TACR2TACR1TACR3CYP2D6HRH1
SCHEMBL8640621 0.86 TACR2 (0.52) TACR2TACR1TACR3CYP2D6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed