SCHEMBL8650818

SCHEMBL8650818

CS(=O)(=O)c1cccc(/C=C(/C(=O)NC(=N)N)c2cccnc2)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.46
VNN1 O95497 1/20 0.42
BRAF P15056 1/20 0.41
F10 P00742 1/20 0.40
AKR1C3 P42330 3/20 0.38
AKR1C2 P52895 1/20 0.38
CYP1A1 P04798 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP1B1 Q16678 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8646691 0.88 CYP1A1 (0.47) NAMPTF10CYP1A1CYP1A2CYP1B1
SCHEMBL8650927 0.86 NPC1 (0.45) NAMPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL8646693 0.85 CYP1A1 (0.42) NAMPTF10CYP1A1CYP1A2CYP1B1
SCHEMBL8646754 0.85 CYP1A1 (0.52) NAMPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL8644166 0.84 CYP1A1 (0.52) F10CYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL8647943 0.83 CYP1A2 (0.47) NAMPTCYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL8646756 0.83 CYP3A4 (0.48) F10AKR1C3CYP1A1CYP1A2CYP1B1
SCHEMBL8650918 0.82 AKR1C3 (0.55) NAMPTAKR1C3AKR1C2PDE4APDE4B
SCHEMBL8650924 0.82 AKR1C3 (0.55) NAMPTAKR1C3AKR1C2PDE4APDE4B
SCHEMBL8648534 0.82 CYP1A1 (0.55) CYP1A1CYP1A2CYP1B1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed