SCHEMBL8655950

SCHEMBL8655950

ClC(Cl)=CCOc1cc(Cl)c(OCCCc2ccc(Cl)cc2)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.37
ALOX15 P16050 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 1/20 0.35
SLC6A2 P23975 2/20 0.34
HRH1 P35367 2/20 0.34
HRH3 Q9Y5N1 2/20 0.34
KCNH2 Q12809 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
CHRM2 P08172 1/20 0.34
ADRA2C P18825 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CACNA1C Q13936 1/20 0.34
SCN5A Q14524 1/20 0.34
CHRM4 P08173 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408013 0.96 IGF1R (0.39) IGF1RALOX15L3MBTL1HTTPPARG
SCHEMBL8518771 0.93 MAOB (0.38) HTTPPARGPPARASLC6A4HTR2C
SCHEMBL8659980 0.90 PPARA (0.39) HTTPPARGPPARAMAPTMAOB
SCHEMBL8659951 0.90 PPARD (0.39) L3MBTL1HTTMAPTMAOBMAOA
SCHEMBL8660296 0.90 HPGD (0.39) L3MBTL1MAOBMAOA
SCHEMBL6548477 0.88 HPGD (0.37) L3MBTL1HTTPPARGPPARAMAPT
SCHEMBL7071500 0.87 NMT1 (0.40) HTTSLC6A2HRH1SLC6A4SLC6A3
SCHEMBL8659996 0.87 FFAR1 (0.36) KCNH2PPARGPPARAMAOBHDAC1
SCHEMBL8405697 0.86 HTT (0.42) HTTHRH3KCNH2
SCHEMBL8408726 0.86 HTT (0.42) HTTHRH3KCNH2PPARAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed