SCHEMBL8656199

SCHEMBL8656199

Cc1ccc(Oc2ccc(Oc3c(C)cc(NC(=O)NC(=O)c4c(F)cccc4Cl)c(C)c3Cl)c(Cl)c2)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 4/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
MAPK1 P28482 1/20 0.39
TLR8 Q9NR97 4/20 0.39
GAA P10253 4/20 0.38
POLB P06746 2/20 0.38
TLR7 Q9NYK1 2/20 0.38
GCGR P47871 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8659740 0.97 MEN1 (0.46) MEN1KMT2ANPSR1MAPTUSP2
SCHEMBL8659386 0.94 NPSR1 (0.43) MEN1KMT2ANPSR1MAPTALDH1A1
SCHEMBL8658960 0.90 KMT2A (0.49) MEN1KMT2ANPSR1MAPTUSP2
SCHEMBL8659850 0.89 MEN1 (0.51) MEN1KMT2ANPSR1MAPTUSP2
SCHEMBL8658863 0.89 MEN1 (0.43) MEN1KMT2ANPSR1MAPTUSP2
SCHEMBL9135134 0.88 MEN1 (0.46) MEN1KMT2ANPSR1MAPTUSP2
SCHEMBL8659373 0.88 NPSR1 (0.43) MEN1KMT2ANPSR1MAPTALDH1A1
SCHEMBL8659368 0.85 GCGR (0.43) KMT2ANPSR1MAPTALDH1A1GCGR
SCHEMBL8659541 0.85 ATM (0.44) MEN1KMT2ANPSR1MAPTALDH1A1
SCHEMBL8659795 0.84 KMT2A (0.49) MEN1KMT2ANPSR1MAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
US-4602109-A Novel pesticidal phenoxyphenyl and phenoxypyridyl benzoyl ureas and process for preparation UNION CARBIDE CORPORATION (US) 1986-07-22 US disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
US-4540578-A Pesticidal phenoxypyridyl benzoyl ureas UNION CARBIDE CORPORATION (US) 1985-09-10 US disclosed
EP-0113247-A1 Pesticidal phenoxyphenyl and phenoxypyridyl benzoyl ureas and process for their preparation UNION CARBIDE CORPORATION (US) 1984-07-11 EP disclosed