Bromide

Bromide

SCHEMBL8660152

Br.Br.c1ccc(P(c2ccccc2)c2ccccc2-c2ccccc2P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
ESR1 P03372 3/20 0.42
ESR2 Q92731 3/20 0.42
DRD1 P21728 2/20 0.41
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1120987 0.97 CYP3A4 (0.58) CYP3A4TDP1ESR1ESR2DRD1
Water SCHEMBL1131329 0.95 CYP3A4 (0.55) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL30350108 0.95 CYP3A4 (0.55) CYP3A4TDP1ESR1ESR2DRD1
Water SCHEMBL1131752 0.95 CYP3A4 (0.55) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL31059891 0.95 CYP3A4 (0.55) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL28427105 0.86 TDP1 (0.46) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL28152680 0.86 TDP1 (0.46) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL29635182 0.85 TDP1 (0.50) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL4004840 0.85 TDP1 (0.50) CYP3A4TDP1ESR1ESR2DRD1
SCHEMBL28333146 0.85 TDP1 (0.50) CYP3A4TDP1ESR1ESR2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5741931-A Phosphepinium salts HOECHST AG (DE) 1998-04-21 US disclosed