SCHEMBL8663399

SCHEMBL8663399

O=C(O)c1cn([C@@H]2C[C@@H]2F)c2c(C(F)(F)F)c(F)c(F)cc2c1=O.O=C(O)c1cn([C@@H]2C[C@@H]2F)c2c(OC(F)F)c(F)c(F)cc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
KCNH2 Q12809 4/20 0.40
TOP2A P11388 4/20 0.39
TOP2B Q02880 4/20 0.39
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 5/20 0.39
HPGD P15428 4/20 0.39
POLB P06746 3/20 0.39
HSD17B10 Q99714 3/20 0.39
OPRM1 P35372 2/20 0.39
PRKD3 O94806 1/20 0.39
ALOX15 P16050 1/20 0.39
CLK2 P49760 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
OPRD1 P41143 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8131420 0.92 TOP2A (0.44) CYP3A4KCNH2TOP2ATOP2BALDH1A1
SCHEMBL8131531 0.92 TOP2A (0.44) CYP3A4KCNH2TOP2ATOP2BALDH1A1
SCHEMBL9094282 0.92 TOP2A (0.44) CYP3A4KCNH2TOP2ATOP2BALDH1A1
SCHEMBL8138702 0.89 TOP2A (0.46) CYP3A4TOP2ATOP2BALDH1A1KDM4E
SCHEMBL9097687 0.89 TOP2A (0.46) CYP3A4TOP2ATOP2BALDH1A1KDM4E
SCHEMBL8137973 0.89 TOP2A (0.46) CYP3A4TOP2ATOP2BALDH1A1KDM4E
SCHEMBL13469793 0.83 CYP3A4 (0.43) CYP3A4KCNH2TOP2ATOP2BALDH1A1
SCHEMBL4747731 0.83 CYP3A4 (0.43) CYP3A4KCNH2TOP2ATOP2BALDH1A1
SCHEMBL8131423 0.81 CYP3A4 (0.33) CYP3A4KCNH2TOP2ATOP2BALDH1A1
SCHEMBL9238212 0.81 CYP3A4 (0.33) CYP3A4KCNH2TOP2ATOP2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5783708-A HEXAHYDROISOINDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1998-07-21 US disclosed