SCHEMBL8665668

SCHEMBL8665668

Cc1cc(C)cc(-c2[nH]c3ccc(N)cc3c2CCNC(=O)OC(C)(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 5/20 0.45
MTNR1A P48039 2/20 0.45
MTNR1B P49286 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8191104 0.88 PPARG (0.51) GNRHR
SCHEMBL6986887 0.87 GNRHR (0.51) GNRHR
SCHEMBL6983015 0.86 CXCR2 (0.55) CYP2C9
SCHEMBL6984508 0.86 GNRHR (0.49) GNRHR
SCHEMBL8185257 0.85 GNRHR (0.49) GNRHRKDM4EALDH1A1
SCHEMBL8668503 0.85 MAPT (0.43) GNRHRMTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL6982073 0.85 GNRHR (0.47) GNRHR
SCHEMBL6983351 0.84 GNRHR (0.51) GNRHR
SCHEMBL8697833 0.83 GNRHR (0.43) GNRHR
SCHEMBL6982574 0.82 GNRHR (0.48) GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871624-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE Merck & Co., Inc. (US) 1998-10-21 EP disclosed
WO-1997021703-A1 ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE MERCK & CO., INC. (US) 1997-06-19 WO disclosed