Bromide

Bromide

SCHEMBL8689149

Br.CCCN(CCC)C1Cc2cc(O)c(O)cc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A known ✓ P08908 1/20 0.56
ADRB2 known ✓ P07550 1/20 0.56
FYN P06241 3/20 0.96
CYP2D6 P10635 2/20 0.62
ALDH1A1 P00352 1/20 0.62
CYP2C9 P11712 1/20 0.62
ALOX15 P16050 1/20 0.62
MAPK1 P28482 1/20 0.62
DRD3 P35462 5/20 0.59
DRD2 P14416 4/20 0.59
LMNA P02545 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
MAPT P10636 1/20 0.59
DRD4 P21917 2/20 0.56
CASP1 P29466 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8443814 0.98 FYN (1.00) FYNCYP2D6ALDH1A1CYP2C9ALOX15
Bromide SCHEMBL7198686 0.89 FYN (0.97) FYNCYP2D6ALDH1A1DRD3DRD2
SCHEMBL29177063 0.88 FYN (0.81) FYNCYP2D6ALDH1A1CYP2C9ALOX15
SCHEMBL22417780 0.87 FYN (0.80) FYNCYP2D6ALDH1A1CYP2C9ALOX15
SCHEMBL10606282 0.86 FYN (1.00) FYNCYP2D6DRD3DRD2LMNA
Bromide SCHEMBL8688813 0.83 DRD3 (0.78) FYNCYP2D6ALDH1A1CYP2C9DRD3
SCHEMBL7090402 0.81 FYN (0.69) FYNCYP2D6ALDH1A1CYP2C9ALOX15
SCHEMBL8693035 0.81 FYN (0.70) FYNCYP2D6ALDH1A1CYP2C9ALOX15
SCHEMBL7449385 0.81 DRD3 (0.78) FYNCYP2D6ALDH1A1CYP2C9DRD3
SCHEMBL27483394 0.80 FYN (0.68) FYNCYP2D6ALDH1A1CYP2C9ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708018-A 2-aminoindans as selective dopamine D3 ligands PHARMACIA & UPJOHN COMPANY (US) 1998-01-13 US disclosed
EP-0712387-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1996-05-22 EP disclosed
WO-1995004713-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS THE UPJOHN COMPANY (US) 1995-02-16 WO disclosed