SCHEMBL8697287

SCHEMBL8697287

CCCCn1c(=O)c2c(ncn2CC[C@H](C)O)n(CCCC)c1=O

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 9/20 0.67
PDE4B Q07343 8/20 0.67
PDE4C Q08493 8/20 0.67
PDE4D Q08499 8/20 0.67
ADORA2A P29274 5/20 0.67
ADORA2B P29275 3/20 0.67
CYP1A2 P05177 2/20 0.53
BLM P54132 2/20 0.53
PMP22 Q01453 2/20 0.53
LMNA P02545 1/20 0.53
ESR1 P03372 1/20 0.53
MAPT P10636 1/20 0.53
NFKB1 P19838 1/20 0.53
ACHE P22303 1/20 0.53
CNOT7 Q9UIV1 4/20 0.53
CYP3A4 P08684 1/20 0.51
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696628 1.00 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL8696632 1.00 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11613478 0.93 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10695023 0.91 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10693202 0.91 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL5606734 0.90 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10808455 0.89 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10694979 0.88 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10694974 0.88 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11611955 0.87 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710272-A INCREASING CEREBRAL BLOOD FLOW HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
EP-0435152-B1 Process for the enantioselective preparation of (omega-1)-hydroxyalkylxanthines HOECHST AG (DE) 1996-11-13 EP disclosed
US-5472873-A Rhodotorula rubra useful in a process for the preparation of (ω-1)-hydroxyalkylxanthines HOECHST AKTIENGESELLSCHAFT (DE) 1995-12-05 US disclosed
US-5310666-A Vascular disorders HOECHST AKTIENGESELLSCHAFT (DE) 1994-05-10 US disclosed
EP-0435152-A2 Process for the enantioselective preparation of (omega-1)-hydroxyalkylxanthines HOECHST AKTIENGESELLSCHAFT (DE) 1991-07-03 EP disclosed