SCHEMBL8697487

SCHEMBL8697487

N#Cc1ccc(C(O)(c2cncnc2)c2cc3ccccc3o2)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.49
CYP3A5 P20815 3/20 0.49
CYP19A1 P11511 13/20 0.48
FNTA P49354 2/20 0.36
FNTB P49356 2/20 0.36
KCNH2 Q12809 1/20 0.35
CYP2A6 P11509 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697501 0.88 CYP19A1 (0.44) CYP3A4CYP3A5CYP19A1FNTAFNTB
SCHEMBL8700871 0.86 CYP3A4 (0.43) CYP3A4CYP3A5CYP19A1KCNH2CYP2A6
SCHEMBL8703062 0.86 CYP19A1 (0.58) CYP3A4CYP3A5CYP19A1
SCHEMBL8696315 0.85 CYP19A1 (0.57) CYP3A4CYP3A5CYP19A1FNTAFNTB
SCHEMBL8697489 0.81 CYP3A4 (0.49) CYP3A4CYP3A5CYP19A1FNTAFNTB
SCHEMBL8696734 0.81 CYP3A4 (0.53) CYP3A4CYP3A5CYP19A1KCNH2
SCHEMBL8698505 0.78 CYP19A1 (0.38) CYP3A4CYP3A5CYP19A1KCNH2CYP2A6
SCHEMBL8697681 0.76 CYP19A1 (0.78) CYP19A1
SCHEMBL8702170 0.76 CYP19A1 (0.43) CYP3A4CYP3A5CYP19A1FNTAFNTB
SCHEMBL8696581 0.76 CYP19A1 (0.65) CYP3A4CYP3A5CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO claimed
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO disclosed