SCHEMBL8710562

SCHEMBL8710562

COC(=O)C1=NNCCC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
CHRM3 P20309 1/20 0.33
TSHR P16473 2/20 0.32
USP2 O75604 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK1 P28482 2/20 0.31
KDM4C Q9H3R0 1/20 0.31
SLC6A2 P23975 1/20 0.30
SPR P35270 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31458552 0.88
SCHEMBL29955988 0.75
SCHEMBL18780818 0.74
SCHEMBL883443 0.69
SCHEMBL1757748 0.69 NPC1 (0.47) L3MBTL1ALDH1A1
SCHEMBL27315111 0.63 GAA (0.53) NPSR1MAPK1KDM4CALDH1A1
SCHEMBL5270576 0.61 NPSR1 (0.35) NPSR1CHRM3TSHRMAPK1KDM4C
SCHEMBL27647692 0.61 CHRM3 (0.44) CHRM3TSHRUSP2L3MBTL1SLC6A2
SCHEMBL5865621 0.61
SCHEMBL4921085 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750690-A HYDROGENATION OF A 1,2-DIALKYLOXO-3-CARBOXY-3-PYRAZOLINE OR 1,2,5,6-TETRAHYDROPYRIDAZINE OR DERIVATIVE; INTERMEDIATES FOR THE HYPOTENSIVE AGENT, ?CILAZAPRIL? HOFFMANN-LA ROCHE INC. (US) 1998-05-12 US disclosed