SCHEMBL8713673

SCHEMBL8713673

CCOC(=O)NC(=N)c1ccc(C(=O)N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)c2ccccc2OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
UBE2N P61088 1/20 0.44
CYP3A4 P08684 2/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA1A P35348 1/20 0.43
LMNA P02545 1/20 0.43
HSD11B1 P28845 1/20 0.43
ALDH1A1 P00352 2/20 0.43
BLM P54132 2/20 0.43
PMP22 Q01453 1/20 0.43
HTT P42858 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL8714573 0.98 CYP2D6 (0.46) CYP2D6CYP2C19KMT2AMEN1UBE2N
SCHEMBL8712283 0.91 CYP2D6 (0.50) CYP2D6CYP2C19KMT2AMEN1CYP3A4
SCHEMBL8710662 0.89 CYP2C19 (0.51) CYP2D6CYP2C19KMT2AMEN1UBE2N
Oxalic Acid SCHEMBL8711032 0.88 CYP2D6 (0.48) CYP2D6CYP2C19KMT2AMEN1CYP3A4
SCHEMBL8711017 0.88 CYP2D6 (0.47) CYP2D6CYP2C19KMT2AMEN1UBE2N
SCHEMBL9232901 0.86 CYP2D6 (0.49) CYP2D6CYP2C19KMT2AMEN1CYP3A4
Oxalic Acid SCHEMBL8716566 0.86 CYP2D6 (0.46) CYP2D6CYP2C19KMT2AMEN1UBE2N
SCHEMBL8711518 0.85 CYP2D6 (0.51) CYP2D6CYP2C19KMT2AMEN1CYP3A4
Fumaric Acid SCHEMBL8710922 0.85 CYP2C19 (0.47) CYP2D6CYP2C19KMT2AMEN1UBE2N
Fumaric Acid SCHEMBL8714316 0.85 CYP2C19 (0.47) CYP2D6CYP2C19KMT2AMEN1UBE2N

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed