SCHEMBL8718367

SCHEMBL8718367

O=c1[nH]ncn1-c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.51
GPR119 Q8TDV5 1/20 0.42
BCHE P06276 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
AR P10275 1/20 0.38
EP300 Q09472 1/20 0.37
KAT2B Q92831 1/20 0.37
ADRB2 P07550 1/20 0.35
NCF1 P14598 1/20 0.35
PLD1 Q13393 1/20 0.35
ALDH1A1 P00352 3/20 0.35
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
CHKA P35790 1/20 0.34
DAO P14920 1/20 0.34
HSD17B10 Q99714 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3518937 0.81 HTT (0.62) HTTGPR119TDP1ALDH1A1HSD17B10
SCHEMBL5906422 0.79 HTT (0.69) HTTGPR119TDP1
SCHEMBL7678192 0.79 HTT (0.47) HTTGPR119TDP1ALDH1A1CCNA2
SCHEMBL7682668 0.78 PDE3B (0.52) HTTLMNA
SCHEMBL1618003 0.78 HTT (0.50) HTTGPR119TDP1ALDH1A1CCNA2
SCHEMBL8718822 0.78 HTT (0.50) HTTGPR119TDP1ALDH1A1KDM4E
SCHEMBL792758 0.78 HTT (0.50) HTTGPR119TDP1ALDH1A1CCNA2
SCHEMBL8718617 0.78 HTT (0.54) HTTGPR119TDP1CCNA2CDK2
SCHEMBL7028939 0.78 HTT (0.50) HTTGPR119TDP1ALDH1A1CCNA2
SCHEMBL21385013 0.74 HTT (0.48) HTTGPR119TDP1ALDH1A1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567982-B1 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-07-01 EP disclosed
US-5466820-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-14 US disclosed
US-5371101-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-06 US disclosed
EP-0567982-A1 Azole compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-11-03 EP disclosed